Efficient Pd-Catalyzed Amination Reactions for Heterocycle Functionalization
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Buchwald_Efficient Pd.pdf
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Author(s) •
Henderson, Jaclyn L.
Buchwald, Stephen Leffler
Date Issued
September 2010
Journal
American Chemical Society (ACS)
Publisher
Organic Letters
Citation
Henderson, Jaclyn L., and Stephen L. Buchwald. “Efficient Pd-Catalyzed Amination Reactions for Heterocycle Functionalization.” Organic Letters 12.20 (2010): 4442–4445.
Version
Author's final manuscript
Abstract
The Pd-catalyzed amination of unprotected benzo-fused heterocycles is reported, which allows for greater flexibility and efficiency in the modification of this important class of molecules. The generality of these simple and efficient procedures is demonstrated through the synthesis of a wide variety of structural types.
MIT Department
Massachusetts Institute of Technology. Department of Chemistry
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DOI of Published Version
https://doi.org/10.1021/ol101929v