Pd-Catalyzed Cross-Coupling Reactions of Amides and Aryl Mesylates
Author(s)Dooleweerdt, Karin; Fors, Brett P.; Buchwald, Stephen Leffler
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A catalyst, based on a biarylphosphine ligand, for the Pd-catalyzed cross-coupling reactions of amides and aryl mesylates is described. This system allows an array of aryl and heteroaryl mesylates to be transformed into the corresponding N-aryl amides in moderate to excellent yields.
DepartmentMassachusetts Institute of Technology. Department of Chemistry
American Chemical Society (ACS)
Dooleweerdt, Karin, Brett P. Fors, and Stephen L. Buchwald. “Pd-Catalyzed Cross-Coupling Reactions of Amides and Aryl Mesylates.” Organic Letters 12.10 (2010): 2350–2353.
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