Efficient Pd-Catalyzed Amination Reactions for Heterocycle Functionalization

Author(s)
Henderson, Jaclyn L.; Buchwald, Stephen Leffler
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Abstract
The Pd-catalyzed amination of unprotected benzo-fused heterocycles is reported, which allows for greater flexibility and efficiency in the modification of this important class of molecules. The generality of these simple and efficient procedures is demonstrated through the synthesis of a wide variety of structural types.
Date issued
2010-09
URI
http://hdl.handle.net/1721.1/71942
Department
Massachusetts Institute of Technology. Department of Chemistry
Journal
American Chemical Society (ACS)
Publisher
Organic Letters
Citation
Henderson, Jaclyn L., and Stephen L. Buchwald. “Efficient Pd-Catalyzed Amination Reactions for Heterocycle Functionalization.” Organic Letters 12.20 (2010): 4442–4445.
Version: Author's final manuscript
ISSN
1523-7060
1523-7052
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