Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids

Author(s)
Niljianskul, Nootaree; DeBergh, John Robbins; Buchwald, Stephen Leffler
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Abstract
A palladium-catalyzed method for the preparation of sulfonamides is described. The process exhibits significant functional group tolerance and allows for the preparation of a number of arylsulfonyl chlorides and sulfonamides under mild conditions.
Date issued
2013-07
URI
http://hdl.handle.net/1721.1/93910
Department
Massachusetts Institute of Technology. Department of Chemistry
Journal
Journal of the American Chemical Society
Publisher
American Chemical Society (ACS)
Citation
DeBergh, J. Robb, Nootaree Niljianskul, and Stephen L. Buchwald. “Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids.” Journal of the American Chemical Society 135, no. 29 (July 24, 2013): 10638–10641.
Version: Author's final manuscript
ISSN
0002-7863
1520-5126
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