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dc.contributor.authorSu, Mingjuan
dc.contributor.authorHoshiya, Naoyuki
dc.contributor.authorBuchwald, Stephen Leffler
dc.date.accessioned2015-04-23T17:16:41Z
dc.date.available2015-04-23T17:16:41Z
dc.date.issued2014-01
dc.date.submitted2013-12
dc.identifier.issn1523-7060
dc.identifier.issn1523-7052
dc.identifier.urihttp://hdl.handle.net/1721.1/96743
dc.description.abstractAn efficient method for the palladium-catalyzed amination of unprotected bromoimidazoles and bromopyrazoles is presented. The transformation is facilitated by the use of our newly developed Pd precatalyst based on the bulky biarylphosphine ligand tBuBrettPhos (L4). The mild reaction conditions employed allow for the preparation of a broad scope of aminoimidazoles and aminopyrazoles in moderate to excellent yields.en_US
dc.description.sponsorshipNational Institutes of Health (U.S.) (Award GM58160)en_US
dc.description.sponsorshipAstellas USA Foundation (Fellowship)en_US
dc.description.sponsorshipJapan Society for the Promotion of Science (Young Scientist Research Fellowship)en_US
dc.language.isoen_US
dc.publisherAmerican Chemical Society (ACS)en_US
dc.relation.isversionofhttp://dx.doi.org/10.1021/ol4035947en_US
dc.rightsArticle is made available in accordance with the publisher's policy and may be subject to US copyright law. Please refer to the publisher's site for terms of use.en_US
dc.sourceAmerican Chemical Societyen_US
dc.titlePalladium-Catalyzed Amination of Unprotected Five-Membered Heterocyclic Bromidesen_US
dc.typeArticleen_US
dc.identifier.citationSu, Mingjuan, Naoyuki Hoshiya, and Stephen L. Buchwald. “Palladium-Catalyzed Amination of Unprotected Five-Membered Heterocyclic Bromides.” Org. Lett. 16, no. 3 (February 7, 2014): 832–835. © 2014 American Chemical Societyen_US
dc.contributor.departmentMassachusetts Institute of Technology. Department of Chemistryen_US
dc.contributor.mitauthorBuchwald, Stephen Leffleren_US
dc.contributor.mitauthorSu, Mingjuanen_US
dc.contributor.mitauthorHoshiya, Naoyukien_US
dc.relation.journalOrganic Lettersen_US
dc.eprint.versionFinal published versionen_US
dc.type.urihttp://purl.org/eprint/type/JournalArticleen_US
eprint.statushttp://purl.org/eprint/status/PeerRevieweden_US
dspace.orderedauthorsSu, Mingjuan; Hoshiya, Naoyuki; Buchwald, Stephen L.en_US
dc.identifier.orcidhttps://orcid.org/0000-0003-3875-4775
mit.licensePUBLISHER_POLICYen_US


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