| dc.contributor.author | Su, Mingjuan | |
| dc.contributor.author | Hoshiya, Naoyuki | |
| dc.contributor.author | Buchwald, Stephen Leffler | |
| dc.date.accessioned | 2015-04-23T17:16:41Z | |
| dc.date.available | 2015-04-23T17:16:41Z | |
| dc.date.issued | 2014-01 | |
| dc.date.submitted | 2013-12 | |
| dc.identifier.issn | 1523-7060 | |
| dc.identifier.issn | 1523-7052 | |
| dc.identifier.uri | http://hdl.handle.net/1721.1/96743 | |
| dc.description.abstract | An efficient method for the palladium-catalyzed amination of unprotected bromoimidazoles and bromopyrazoles is presented. The transformation is facilitated by the use of our newly developed Pd precatalyst based on the bulky biarylphosphine ligand tBuBrettPhos (L4). The mild reaction conditions employed allow for the preparation of a broad scope of aminoimidazoles and aminopyrazoles in moderate to excellent yields. | en_US |
| dc.description.sponsorship | National Institutes of Health (U.S.) (Award GM58160) | en_US |
| dc.description.sponsorship | Astellas USA Foundation (Fellowship) | en_US |
| dc.description.sponsorship | Japan Society for the Promotion of Science (Young Scientist Research Fellowship) | en_US |
| dc.language.iso | en_US | |
| dc.publisher | American Chemical Society (ACS) | en_US |
| dc.relation.isversionof | http://dx.doi.org/10.1021/ol4035947 | en_US |
| dc.rights | Article is made available in accordance with the publisher's policy and may be subject to US copyright law. Please refer to the publisher's site for terms of use. | en_US |
| dc.source | American Chemical Society | en_US |
| dc.title | Palladium-Catalyzed Amination of Unprotected Five-Membered Heterocyclic Bromides | en_US |
| dc.type | Article | en_US |
| dc.identifier.citation | Su, Mingjuan, Naoyuki Hoshiya, and Stephen L. Buchwald. “Palladium-Catalyzed Amination of Unprotected Five-Membered Heterocyclic Bromides.” Org. Lett. 16, no. 3 (February 7, 2014): 832–835. © 2014 American Chemical Society | en_US |
| dc.contributor.department | Massachusetts Institute of Technology. Department of Chemistry | en_US |
| dc.contributor.mitauthor | Buchwald, Stephen Leffler | en_US |
| dc.contributor.mitauthor | Su, Mingjuan | en_US |
| dc.contributor.mitauthor | Hoshiya, Naoyuki | en_US |
| dc.relation.journal | Organic Letters | en_US |
| dc.eprint.version | Final published version | en_US |
| dc.type.uri | http://purl.org/eprint/type/JournalArticle | en_US |
| eprint.status | http://purl.org/eprint/status/PeerReviewed | en_US |
| dspace.orderedauthors | Su, Mingjuan; Hoshiya, Naoyuki; Buchwald, Stephen L. | en_US |
| dc.identifier.orcid | https://orcid.org/0000-0003-3875-4775 | |
| mit.license | PUBLISHER_POLICY | en_US |
| mit.metadata.status | Complete | |
