Structural and biophysical insights into the mode of covalent binding of rationally designed potent BMX inhibitors
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<p>We identified potent, functionalisable BMX inhibitors and revealed their covalent mode of binding to BMX by X-ray crystallography.</p>
Date issued
2020-08Department
Koch Institute for Integrative Cancer Research at MITJournal
RSC Chemical Biology
Publisher
Royal Society of Chemistry (RSC)
Citation
Seixas, João D, Sousa, Bárbara B, Marques, Marta C, Guerreiro, Ana, Traquete, Rui et al. 2020. "Structural and biophysical insights into the mode of covalent binding of rationally designed potent BMX inhibitors." RSC Chemical Biology, 1 (4).
Version: Final published version
ISSN
2633-0679